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High-Throughput Drug Screening Facility
Publications
Veach DR, Namavari M, Beresten, Balatoni TJ, Minchenko M, Djaballah H, Finn RD, Clarkson B, Gelovani JG, Bornmann, WG and Larson SM (2005) "Synthesis and in vitro examination of [124I]-, [125I]- and [131I]-2-(4-iodophenylamino) pyrido[2,3-d]pyrimidin-7-one radiolabeled Abl kinase inhibitors" Nuclear Medicine and Biology 32:313-321.
Antczak, C, Shum, D, Escobar, S, Bassit, B, Kim, E, Venkatraman, E, Wu, N, Yang, G, Ouerfelli, O, Li, Y, Scheinberg, DA, Djaballah, H (2007) "High-throughput Identification of Inhibitors of the Cancer Target Human Mitochondrial Peptide Deformylase" J Biomol Screen 12:521-535.
Ramajayam R, Gididhar, R, Yadav, MR, Djaballah H, Shum, D, Radu, C (2007) "Synthesis and antiproliferative activity of some diaryldiazepines and diarylpyrimidines" J Enz Inhib Med Chem 22:716-721.
Veach DR, Namavari M, Pillarsetty N, Santos EB, Beresten-Kochetkov T, Lambek C, Punzalan BJ, Antczak C, Smith-Jones PM, Djaballah H, Clarkson B, Larson SM (2007) "Synthesis and biological evaluation of a fluorine-18 derivative of dasatinib" J Med Chem 50:5853-5857.
Deng L, Dai P, Ciro A, Smee DF, Djaballah H, Shuman S (2007) "Identification of novel antipoxviral agents: Mitoxantrone inhibits vaccinia virus replication by blocking virion assembly" J Virology 81:13392-402.
Ramajayam R, Gididhar, R, Yadav, MR, Balaraman R, Djaballah H, Shum, D, Radu, C (2008) "Synthesis, antileukemic and antiplatelet activities of 2,3-diaryl-6,7-dihydro-5H-1,4-diazepines" Eur J Med Chem 43:2004-10.
Shum D, Radu C, Kim E, Cajuste M, Shao Y, Seshan V.E., Djaballah H (2008) "A high density assay format for the detection of novel cytotoxic agents in large chemical libraries" J Enz Inhib Med Chem 23:931-45.
Eckelbarger JD, Wilmot JT, Epperson MT, Thakur CS, Shum D, Antczak C, Tarassishin L, Djaballah H, Gin DY (2008) "Synthesis of Antiproliferative Cephalotaxus Esters and Their Evaluation against Several Human Hematopoietic and Solid Tumor Cell Lines: Uncovering Differential Susceptibilities to Multi-Drug Resistance" Chem Eur J 14:1-15
Antczak C, Radu C, Djaballah H (2008) "A Profiling Platform for the Identification of Selective Metalloprotease Inhibitors" J Biomol Screen 13:285-294
Desbordes SC, Placantonakis DG, Ciro A, Socci ND, Lee G, Djaballah H, Studer L (2008) High-throughput screening assay for the identification of compounds regulating self-renewal and differentiation in human embryonic stem cells Cell Stem Cell 2:602-12.
Antczak C, Kloepping C, Radu C, Genski T, Muller-Kuhrt L, Siems K, de Stanchina E, Abramson DH, Djaballah H (2009) "Revisiting Old Drugs as Novel Agents for Retinoblastoma: In vitro and In vivo Antitumor Activity of Cardenolides" Invest Ophthalmol Vis Sci (in press)
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